Cirewar Corydalis Tetrahydropalmatine (dl-THP)
Tetrahydropalmatine (THP), wanda aka fi sani da dl-THP, Corydalin hydrochloride, ko kuma Corydalin Tube Extract, wani sinadari ne da aka rarraba a matsayin isoquinoline alkaloid. Ana cire shi daga tuber na ganyen kasar Sin Corydalis yanhusuo. THP wani abu ne mai launin crystalline mara launi ko rawaya mai haske tare da ɗanɗano mai ɗaci da kuma wurin narkewa na 147-149°C. Ba ya narkewa a cikin ruwa amma yana narkewa sosai a cikin ether, chloroform, da ethanol. Gishirin hydrochloride da sulfate suna narkewa a cikin ruwa.
An yi nazarin THP game da tasirin magunguna daban-daban, ciki har da tasirinsa na rage zafi, maganin sa barci, kariya daga jijiyoyi, hana platelet, hana gyambon ciki, hana ciwan ciki, da kuma hana shan kwayoyi. Ana kyautata zaton yana da tasirin rage zafi ta hanyar daidaita ayyukan masu karɓar dopamine na tsakiya kuma ya nuna yuwuwar kare jijiyoyi daga raunin ischemic. Bugu da ƙari, THP ta nuna tasirin haɗa platelet kuma an bincika yuwuwarta wajen magance gyambon ciki, hana haɓakar ƙwayoyin ƙari, da kuma taimakawa wajen shan ƙwayoyi.
Gabaɗaya, Tetrahydropalmatine (dl-THP) wani sinadari ne mai nau'ikan kaddarorin magani kuma an yi bincike mai zurfi kan yuwuwar amfani da shi wajen magance cututtuka. Don ƙarin bayani tuntuɓigrace@biowaycn.com.
Ga siffofin samfurin Tetrahydropalmatine (THP) tare da fa'idodin lafiyarsu:
1. Abubuwan da ke rage radadi:THP yana nuna tasirin rage zafi ta hanyar daidaita ayyukan masu karɓar dopamine na tsakiya, yana ba da sauƙin rage zafi ba tare da yuwuwar jaraba mai mahimmanci ba.
2. Tasirin Kare Jijiyoyi:THP ta nuna yuwuwar kare jijiyoyi daga raunin ischemic, rage apoptosis na jijiyoyi, da kuma rage matakan glutamate a cikin kwakwalwa, wanda hakan na iya taimakawa wajen kare lafiyar jijiyoyi.
3. Tarin magungunan hana platelet:An gano cewa THP yana hana tarawar platelets, wanda hakan ke rage haɗarin kamuwa da gudan jini da kuma abubuwan da suka shafi zuciya da jijiyoyin jini.
4. Tallafin Lafiyar Ciki:THP ya nuna tasirin hana gyambon ciki kuma yana iya taimakawa wajen rage fitar da sinadarin acid na ciki, yana ba da sauƙi daga gyambon ciki da sauran cututtuka masu alaƙa.
5. Yiwuwar Aikin Maganin Ƙwayar Cutar:THP ya nuna tasirin cytotoxic akan ƙwayoyin ƙari, yana nuna yuwuwar rawa wajen hana ci gaban ƙari.
6. Halayen Yaƙi da Shan Kwaya:An yi nazarin THP game da yuwuwar rage alamun janyewar da ke da alaƙa da jarabar opioid da abubuwan ƙarfafawa, yana ba da alƙawarin maganin jaraba da rigakafin sake dawowa.
Waɗannan fasalulluka suna nuna fa'idodi daban-daban na lafiya da kuma yuwuwar amfani da Tetrahydropalmatine (THP) wajen magance cututtuka.
Tetrahydropydalin (dl-THP) na cikin alkaloids na isoquinoline kuma alkaloid ne, galibi a cikin nau'in Corydalis lucidum (Yan Hu Suo), amma kuma a cikin wasu tsire-tsire kamar Stephania rotunda. Waɗannan tsire-tsire suna da amfani na gargajiya a cikin maganin ganye na ƙasar Sin.Corydalis shuka ce mai tsiro mai tsiro na dindindin, tsayinta daga santimita 10 zuwa 20, tana da busassun ganye masu siffar ƙwallo. Tushenta na sama da ƙasa gajeru ne kuma siriri, tare da sikelin sama da tushe. Ganyen basal da ganyen cauline suna kama da juna a siffarsu, tare da busassun ganye; ganyen cauline suna canzawa, tare da ganyen hade 2 da 3. Ganyen na biyu galibi ba ya rabuwa cikakke kuma yana da lobe mai zurfi. Ƙananan ganyen suna da tsayi, oval, ko oval. Linear, kimanin santimita 2 tsayi, tare da kololuwar da ba ta da kaifi ko kaifin gani da gefuna masu kyau. Furen furanninsa suna da siffar raceme, tare da ganyen ƙarshe ko akasin haka; bracts suna da faɗi lanceolate; furanni suna da ja-shunayya kuma suna girma a kwance akan siraran pedicels, waɗanda tsawonsu ya kai milimita 6; calyx yana faɗuwa da wuri; furannin suna da 4 kuma whorls na waje suna da 2. Rassa sun ɗan fi girma, tare da gefuna ruwan hoda da tsakiyar shuɗi-shunayya. Akwai sashe ɗaya na sama, kuma wutsiyar ta faɗa zuwa dogon spur. Tsawon spur ya kai kusan rabin jimlar tsawon. Sassan ciki guda biyu sun fi ƙanƙanta fiye da sassan waje guda biyu. Ƙarshen sama yana da shuɗi-shuɗi kuma an warke, kuma ɓangaren ƙasan yana da ruwan hoda; Stamens ɗin guda 6 ne, kuma an haɗa filaments ɗin zuwa guda biyu, kowannensu yana da anthers guda 3; kwai yana da lebur-cylindrical, salon yana da gajere kuma siriri, kuma ƙazanta shine 2, kamar ƙaramin malam buɗe ido. 'Ya'yan itacensa ƙasfa ne. Ana samar da Corydalis galibi a tsaunuka ko ciyayi. Manyan yankunan da ake samar da su sun haɗa da Zhejiang, Hebei, Shandong, Jiangsu, da sauran wurare.
| Bincike | Ƙayyadewa |
| Gwaji | Tetrahydropalmatine ≥98% |
| Bayyanar | Foda mai haske rawaya zuwa fari Foda |
| Toka | ≤0.5% |
| Danshi | ≤5.0% |
| Magungunan kashe kwari | Mara kyau |
| Karfe masu nauyi | ≤10ppm |
| Pb | ≤2.0ppm |
| As | ≤2.0ppm |
| Ƙamshi | Halaye |
| Girman ƙwayoyin cuta | Ramin 100% zuwa 80 |
| Kwayoyin cuta: | |
| Jimlar ƙwayoyin cuta | ≤1000cfu/g |
| Fungi | ≤100cfu/g |
| Salmgosella | Mara kyau |
| Coli | Mara kyau |
Ga masana'antun aikace-aikacen samfuran Tetrahydropalmatine (THP):
1. Magunguna:Ana amfani da THP a masana'antar magunguna don haɓaka magungunan rage radadi da magungunan kariya daga jijiyoyi.
2. Sinadaran Abinci Mai Gina Jiki:Ana amfani da THP a masana'antar abinci mai gina jiki don ƙirƙirar kari wanda ke nufin rage zafi da tallafin lafiyar ciki.
3. Fasahar kere-kere:THP ta gano aikace-aikace a fannin fasahar kere-kere don bincike kan hanyoyin magance platelet da kuma yiwuwar maganin cutar kansa.
4. Kula da Lafiya:An haɗa THP a cikin samfuran kiwon lafiya don magance jaraba da alamun janyewa da ke da alaƙa da amfani da opioid da abubuwan ƙarfafawa.
5. Kayan kwalliya:Ana binciken THP a fannin kayan kwalliya don yuwuwar lafiyar fata da aikace-aikacen hana kumburi.
Waɗannan masana'antu suna nuna nau'ikan amfani da Tetrahydropalmatine (THP) a fannoni daban-daban na haɓaka samfura da bincike.
Ana ƙera Kayayyakinmu ta amfani da tsauraran matakan kula da inganci kuma suna bin ƙa'idodi masu girma na tsarin samarwa. Muna ba da fifiko ga aminci da ingancin samfurinmu, muna tabbatar da cewa ya cika buƙatun ƙa'idoji da takaddun shaida na masana'antu. Wannan alƙawarin ga inganci yana nufin tabbatar da aminci da amincewa ga ingancin samfurinmu. Tsarin samarwa gabaɗaya shine kamar haka:
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